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2015

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·  62. "Regio-, Diastereo-, and Enantioselective Nitroso-Diels–Alder Reaction of 1, 3-Diene-1-carbamates Catalyzed by Chiral Phosphoric Acids"

Pous, J.; Courant, T.; Bernadat, G.; Iorga, B.I.; Blanchard, F.; Masson, G. J. Am. Chem. Soc., 2015, 137, 11950-11953. DOI 10.1021/jacs.5b08515 Synfacts, 2015, 11, 1212.

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·  61. "Three-Component Photoredox-Mediated Chloro-, Bromo-, or Iodotrifluoromethylation of Alkenes"

Carboni, A.; Dagousset, G.; Magnier, E.; Masson, G. Synthesis, 2015, 47, 2439- 2445. DOI 10.1055/s-0034-1378715

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·  60. "Formal Asymmetric Organocatalytic [3 + 2] Cyclization between Enecarbamates and 3-Indolylmethanols – a Rapid Access to 3-Aminocyclopenta[b]indoles"

Lebée, C.; Kataja, A. O.; Blanchard, F.; Masson, G. Chem. Eur. J., 2015, 21, 8399-8402. DOI 10.1002/chem.201500749

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·  59. "Enamide derivatives: Versatile Building Blocks for Total Synthesis"

Courant, T.; Dagousset, G.; Masson, G., Synthesis, 2015, 47, 1799-1856. DOI 10.1055/s-0034-1378706

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·  58. "Catalytic, highly enantioselective, direct amination of enecarbamates"

Dumoulin, A.; Lalli, C.; Retailleau, P.; Masson, G. Chem. Commun., 2015, 51, 5383-5386. DOI 10.1039/C4CC08052A

 

2014

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·  57. "Enamide derivatives: Versatile Building Blocks for Highly Functionalized α,β-Substituted Amines"

Bernadat, G.; Masson, G. Synlett, 2014, 25, 2842-2867. DOI 10.1055/s-0034-1379166

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·  56. "Chiral Calcium-BINOL Phosphate Catalyzed Diastereo- and Enantioselective Synthesis of syn-1,2-Disubstituted 1,2-Diamines: Scope and Mechanistic Studies"

Lalli, C.; Dumoulin, A.; Lebée, C.; Drouet, F.; Guérineau, V.; Touboul, D.; Gandon, V.; Zhu, J.; Masson, G. Chem. Eur. J., 2014, 21, 1704-1712. DOI 10.1002/chem.201405286

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·  55. "Imine and iminium precursors as versatile intermediates in enantioselective organocatalysis"

Kataja, A. O.; Masson, G. Tetrahedron, 2014, 70, 8783-8815. DOI 10.1016/j.tet.2014.06.101

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·  54. "One pot and selective intermolecular aryl- and heteroaryltrifluoromethylation of alkenes by photoredox catalysis"

Carboni, A.; Dagousset, G.; Magnier, E.; Masson, G. Chem. Commun., 2014, 50, 14197-14200. DOI 10.1039/C4CC07066F

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·  53. "Photoredox-induced three-component azido- and aminotrifluoromethylation of alkenes"

Dagousset, G.; Carboni, A.; Magnier, E.; Masson, G. Org. Lett., 2014, 16, 4340-4343. DOI 10.1021/ol5021477

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·  52. "Phosphoric Acid Catalyzed Diastereo- and Enantioselective Synthesis of Substituted 1,3-Diaminotetralins"

Dagousset, G.; Erb, W.; Zhu, J.; Masson, G. Org. Lett., 2014, 16, 2554-2557. DOI 10.1021/ol500946w

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·  51. "Cerium(IV) Ammonium Nitrate Mediated Three-Component α-Allylation of Imine Surrogates"

Bekkaye, M.; Masson, G. Org. Lett., 2014, 16, 1510-1513. DOI 10.1021/ol5004143

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·  50. "Photoredox-Induced Three-Component Oxy-, Amino-, and Carbotrifluoro-methylation of Enecarbamates"

Carboni, A.; Dagousset, G.; Magnier, E.; Masson, G. Org. Lett., 2014, 16, 1240-1243. DOI 10.1021/ol500374e

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·  49. "NIS-Assisted Aza-Friedel–Crafts Reaction with α-Carbamoysulfides as Precursors of N-Carbamoylimines"

George, N.; Bekkaye, M.; Alix, A.; Zhu, J.; Masson, G. Chem. Eur. J., 2014, 20, 3621-3625. DOI 10.1002/chem.201400117

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·  48. "An Asymmetric Three-Component Povarov Reaction: Synthesis of tetrahydropyrrolo[3,2-b]pyridines or tetrahydropyrazolo[4,3-b]pyridines"

Brioche, J.; Courant, T.; Alcaraz, L.; Stocks, M.; Furber, M.; Zhu, J.; Masson, G. Adv. Synth. Catal., 2014, 356, 1719-1724. DOI 10.1002/adsc.201400093

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2013

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·  47. "Iron Chloride-Catalyzed Three-Component Domino Sequences: Syntheses of Functionalized α-Oxy-N-acylhemiaminals and α-Oxyimides"

Drouet, F.; Zhu, J.; Masson, G. Adv. Synth. Cat., 2013, 355, 3563-3569. DOI 10.1002/adsc.201300847

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·  46. "Highly Enantioselective Aza-Diels–Alder Reaction of 1-Azadienes with Enecarbamates Catalyzed by Chiral Phosphoric Acids"

He, L.; Laurent, G.; Retailleau, P.; Folléas, B.; Brayer, J.-L.; Masson, G. Angew. Chem. Int. Ed., 2013, 52, 11088-10091. Synfacts, 2013, 10, 1235. DOI 10.1002/ange.201304969

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·  45. "Ugi Four-Component Reaction of Alcohols: Stoichiometric and Catalytic Oxidation/MCR Sequences"

Drouet, F.; Masson, G.; Zhu, J. Org. Lett., 2013, 15, 2854-2857. DOI 10.1021/ol401181a

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·  44. "Metal-Free Dioxygenation of Enecarbamates Mediated by a Hypervalent Iodine Reagent"

Bekkaye, M.; Su, Y.; Masson, G. Eur. J. Org. Chem., 2013, 3978-3982. DOI 10.1002/ejoc.201300501

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·  43. "Chiral Phosphoric Acid-Catalyzed Enantioselective Aza-Friedel-Crafts Alkylation of Indoles with γ-Hydroxy-γ-lactams"

Courant, T.; Kumarn, S.; He, L.; Masson, G. Adv. Synth. Catal., 2013, 355, 836-840. DOI 10.1002/adsc.201201008

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·  42. “Catalytic enantioselective [4 + 2]-cycloaddition: a strategy to access aza-hexacycles”

Masson, G.; Lalli, C.; Benohoud, M.; Dagousset, G. Chem. Soc. Rev., 2013, 42, 902-923. DOI 10.1039/C2CS35370A

 

2012

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·  41. "Organocatalytic Enantioselective One-pot Four-component Ugi-type Multicomponent Reaction for the Synthesis of Epoxy-tetrahydropyrrolo[3,4-b]pyridin-5-ones"

Su, Y.; Bouma, M. J.; Alcarez, L.; Stocks, M.; Furber, M.; Masson, G.; Zhu, J. Chem. Eur. J., 2012, 18, 12624-12627. DOI doi.org/10.1002/chem.201202174

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·  40. "Amidation of Aldehydes and Alcohols via α-Iminonitriles and a Sequential Oxidative Three-component Strecker Reaction/Thio-Michael Addition/Alumina-promoted Hydrolysis to Access α-Mercaptoamides from Aldehydes, Amines and Thiols"

Gualtierotti, J.-B.; Schumacher, X.; Fontaine, P.; Masson, G.; Wang, Q.; Zhu, J. Chem. Eur. J., 2012, 18, 14812-14819. DOI 10.1002/chem.201202291

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·  39. "Highly Enantioselective Electrophilic α-Bromination of Enecarbamates: Chiral Phosphoric Acid and Calcium Phosphate Salt Catalysts"

Allix, A.; Lalli, C.; Retailleau, P.; Masson, G. J. Am. Chem. Soc., 2012, 134, 10389-10392. DOI 10.1021/ja304095z Synfacts, 2012, 9, 1023.

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·  38. "Chiral Phosphoric Acid Catalyzed Inverse-Electron-Demand Aza-Diels–Alder Reaction of Isoeugenol Derivatives"

He, L.; Bekkaye, M.; Retailleau, P.; Masson, G. Org. Lett., 2012, 14, 3158-3161. DOI 10.1021/ol301251h

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·  37. "Chiral Phosphoric Acid-Catalyzed Enantioselective Three-Component Povarov Reaction Using Cyclic Enethioureas as Dienophiles: Stereocontrolled Access to Enantioenriched Hexahydropyrroloquinolines"

Dagousset, G.; Retailleau, P.; Masson, G.; Zhu, J. Chem. Eur. J., 2012, 18, 5869-5873. DOI 10.1002/chem.201200523

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·  36. "Exploiting the Divergent Reactivity of Isocyanoacetates: One-Pot Three-Component Synthesis of Functionalized Angular Furoquinolines"

Bouma, M. J.; Bonne, D.; Masson, G.; Zhu, J. Eur. J. Org. Chem., 2012, 475-479. DOI 10.1002/ejoc.201101567

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·  35. "Photoredox Initiated α-Alkylation of Imines via a Three-Component Radical/Cationic Reaction"

Courant, T. Masson, G. Chem. Eur. J., 2012, 18, 423-427. DOI 10.1002/chem.201103062

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2011

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·  34. "Catalytic Enantioselective Cycloaddition with Chiral Lewis Bases"

Lalli, C.; Brioche, J.; Bernadat, G.; Masson, G. Curr. Org. Chem., 2011, 15, 4108-4127. DOI 10.2174/138527211798109178

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·  33. "Chiral Phosphoric Acid-Catalyzed Enantioselective Three-Component Povarov Reaction Using Enecarbamates as Dienophiles: Highly Diastereo- and Enantioselective Synthesis of Substituted 4-Aminotetrahydroquinolines"

Dagousset, G.; Zhu, J.; Masson, G. J. Am. Chem. Soc., 2011, 133, 14804-14813. DOI 10.1021/ja205891m

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·  32. "A practical, one-pot multicomponent synthesis of α-amidosulfides and its application as latent N-acylimines in Friedel-Crafts reaction"

George, N.; Bekkaye, M.; Masson, G.; Zhu, J. Eur. J. Org. Chem., 2011, 3695-3699.  DOI 10.1002/ejoc.201100426

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·  31. "Cinchona Alkaloid-Amides catalyzed Enantioselective Formal [2 + 2] Cycloadditions of Allenoates and imines: Enantioselective Synthesis of 2,4-Substituted Azetidines"

Denis, J. B.;  Masson,  G.; Retailleau, P.; Zhu, J. Angew. Chem. Int. Ed., 2011, 50, 5356-5360. DOI 10.1002/ange.201100706 Synfacts, 2011, 8, 792.

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·  30. "Asymmetric Synthesis of 2,4,6-Trideoxy-4-(dimethylamino)-3-C-methyl-L-lyxohexopyranose (Lemonose)"

Bernadat, G.; George, N.; Couturier, C.; Masson, G.; Schlama, T.; Zhu, J. Synlett, 2011, 576-578. DOI 10.1055/s-0030-1259531

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·  29. "Chiral Calcium Organophosphate-Catalyzed Enantioselective Electrophilic Amination of Enamides"

Drouet, F.; Lalli, C.; Liu, H.; Masson, G.; Zhu, J. Org. Lett., 2011, 13, 94-97. DOI 10.1021/ol102625s

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·  28. "Exploiting the Divergent Reactivity α-Isocyanoacetate: Multicomponent Synthesis of 5-Alkoxyoxazole and Heterocycles Thereof" Lalli, C.; Bouma, M. J.; Bonne, D.; Masson, G.; Zhu, J. Chem. Eur. J., 2011, 17, 880-889. DOI 10.1002/chem.201002098

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